SCHEMBL6987136

SCHEMBL6987136

Clc1cccc(NCCCCN2CCN3CCCCC3C2)c1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.50
HTR7 P34969 3/20 0.46
POLB P06746 1/20 0.46
HRH3 Q9Y5N1 1/20 0.42
KDR P35968 1/20 0.42
CCR2 P41597 1/20 0.42
KCNH2 Q12809 1/20 0.42
MCHR1 Q99705 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5842025 0.99 SIGMAR1 (0.49) SIGMAR1HTR7POLBHRH3KDR
SCHEMBL5842369 0.90 SIGMAR1 (0.50) SIGMAR1HTR7POLB
Hydrochloric Acid SCHEMBL5840938 0.89 SIGMAR1 (0.49) SIGMAR1HTR7POLB
SCHEMBL6987164 0.87 SIGMAR1 (0.46) SIGMAR1HTR7
SCHEMBL5841805 0.87 SIGMAR1 (0.61) SIGMAR1HTR7HRH3CCR2KCNH2
Hydrochloric Acid SCHEMBL5841049 0.86 SIGMAR1 (0.49) SIGMAR1HTR7HRH3MCHR1
Hydrochloric Acid SCHEMBL5841184 0.86 SIGMAR1 (0.46) SIGMAR1HTR7
Hydrochloric Acid SCHEMBL5842691 0.86 SIGMAR1 (0.60) SIGMAR1HTR7HRH3CCR2KCNH2
SCHEMBL6983319 0.82 ALDH1A1 (0.57) POLBCCR2KCNH2MCHR1
SCHEMBL6985304 0.81 SIGMAR1 (0.46) SIGMAR1HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed