SCHEMBL6987380

SCHEMBL6987380

Cc1cccc(CNC(=O)N2CCN(C(=O)SC(=O)c3ccccc3)CC2)c1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTDSP1 Q9GZU7 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
KDM4E B2RXH2 1/20 0.50
LMNA P02545 2/20 0.49
FAAH O00519 1/20 0.49
P2RY12 Q9H244 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 1/20 0.47
ASAH1 Q13510 2/20 0.46
METAP2 P50579 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
PKM P14618 1/20 0.45
TP53 P04637 2/20 0.44
HTT P42858 1/20 0.44
RECQL P46063 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TPSAB1 Q15661 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6987696 0.99 CTDSP1 (0.56) CTDSP1TDP1KDM4ELMNAFAAH
SCHEMBL6987979 0.88 KDM4E (0.59) CTDSP1TDP1KDM4ELMNAMEN1
Hydrochloric Acid SCHEMBL6991722 0.87 KDM4E (0.58) CTDSP1TDP1KDM4ELMNAMEN1
SCHEMBL6991815 0.81 ALDH1A1 (0.52) KDM4ELMNAP2RY12MEN1KMT2A
SCHEMBL6992011 0.80 PKM (0.59) KDM4EFAAHMEN1KMT2AHRH3
Hydrochloric Acid SCHEMBL6990747 0.80 ALDH1A1 (0.51) KDM4ELMNAP2RY12MEN1KMT2A
Hydrochloric Acid SCHEMBL6989166 0.79 PKM (0.58) KDM4EFAAHMEN1KMT2AHRH3
Hydrochloric Acid SCHEMBL6990408 0.78 KMT2A (0.51) KDM4EFAAHMEN1KMT2AHTT
SCHEMBL29313543 0.76 CHRM3 (0.56) CTDSP1TDP1KDM4ELMNAFAAH
SCHEMBL6987336 0.75 CNR1 (0.59) TDP1KDM4EMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343775-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-09-17 EP disclosed
WO-2002048124-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-20 WO disclosed