SCHEMBL6992011

SCHEMBL6992011

COc1ccc(CNC(=O)N2CCN(C(=O)SC(=O)c3ccccc3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.59
GLA P06280 1/20 0.54
HRH3 Q9Y5N1 2/20 0.54
NPC1 O15118 4/20 0.51
GFER P55789 1/20 0.51
KDM4E B2RXH2 2/20 0.50
TSHR P16473 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
FAAH O00519 1/20 0.49
MMP1 P03956 1/20 0.48
MMP3 P08254 1/20 0.48
MMP7 P09237 1/20 0.48
MMP9 P14780 1/20 0.48
MMP13 P45452 1/20 0.48
RAB9A P51151 1/20 0.48
RYR2 Q92736 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6989166 0.99 PKM (0.58) PKMGLAHRH3NPC1GFER
SCHEMBL6987979 0.88 KDM4E (0.59) HRH3KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL6991722 0.87 KDM4E (0.58) HRH3KDM4EMEN1KMT2A
SCHEMBL6991958 0.83 MAPT (0.67) NPC1TSHRMEN1KMT2AFAAH
Hydrochloric Acid SCHEMBL6989666 0.82 MAPT (0.65) NPC1TSHRMEN1KMT2AFAAH
SCHEMBL6987380 0.80 CTDSP1 (0.57) PKMHRH3KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL6987696 0.79 CTDSP1 (0.56) PKMHRH3KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL6990408 0.78 KMT2A (0.51) KDM4ETSHRMEN1KMT2AFAAH
SCHEMBL6991815 0.78 ALDH1A1 (0.52) PKMKDM4EMEN1KMT2A
SCHEMBL5466489 0.78 MEN1 (0.72) PKMGLAHRH3NPC1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343775-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-09-17 EP disclosed
WO-2002048124-A2 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-06-20 WO disclosed