SCHEMBL6987431

SCHEMBL6987431

O=C(c1ccc(OCc2ccccc2Cl)cc1)N1CCCCc2sccc21

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 7/20 0.60
AVPR1B P47901 5/20 0.60
NR4A2 P43354 1/20 0.50
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
AVPR2 P30518 8/20 0.48
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 2/20 0.44
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44
OXTR P30559 5/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6988048 0.85 NAAA (0.55) AVPR1AAVPR1BNR4A2AVPR2ALDH1A1
SCHEMBL6986447 0.80 AVPR1A (0.71) AVPR1AAVPR1BAVPR2
SCHEMBL7093443 0.79 ALDH1A1 (0.58) AVPR1AAVPR1BAVPR2ALDH1A1MAPT
SCHEMBL6991585 0.76 AVPR1A (0.50) AVPR1AAVPR1BAVPR2ALDH1A1MAPT
SCHEMBL4146200 0.76 AVPR1A (0.68) AVPR1AAVPR1BAVPR2HPGDOXTR
SCHEMBL6991806 0.76 AVPR1A (0.47) AVPR1AAVPR1BAVPR2ALDH1A1MAPT
SCHEMBL6991852 0.76 AVPR1A (0.49) AVPR1AAVPR1BAVPR2ALDH1A1MAPT
SCHEMBL6988528 0.75 AVPR1A (1.00) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL6989910 0.75 AVPR1A (0.46) AVPR1AAVPR1BAVPR2ALDH1A1MAPT
SCHEMBL6202224 0.74 AVPR1A (0.54) AVPR1AAVPR1BAVPR2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811008-B1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS WYETH CORP (US) 2003-10-01 EP disclosed