SCHEMBL6987545

SCHEMBL6987545

CCCCOc1ccc([S+]([O-])N2CC(NCc3ccccc3)C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.43
CYP2C9 P11712 2/20 0.43
LTA4H P09960 3/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
RORC P51449 1/20 0.37
LMNA P02545 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
S1PR1 P21453 1/20 0.37
S1PR5 Q9H228 1/20 0.37
BCHE P06276 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983340 0.77 ADRB3 (0.59) MEN1KMT2AMAPTADRB2ADRB1
SCHEMBL6985385 0.72 ADRB3 (0.47) MEN1KMT2ALMNAMAPTADRB2
SCHEMBL6980419 0.72 KMT2A (0.55) HRH3CYP2C9MEN1KMT2AMAPT
SCHEMBL5555203 0.72 HRH3 (0.58) HRH3CYP2C9MEN1KMT2ARAB9A
SCHEMBL3268536 0.69 KDM1A (0.68)
SCHEMBL14313486 0.67 HRH3 (0.42) HRH3LTA4HNPC1RAB9AHPGD
SCHEMBL425903 0.65 LTA4H (0.63) HRH3CYP2C9LTA4HLMNACYP1A2
SCHEMBL3212615 0.65 LTA4H (0.63) HRH3CYP2C9LTA4HLMNACYP1A2
SCHEMBL9965855 0.65 ACHE (0.54) MEN1KMT2ARAB9ABCHEACHE
SCHEMBL16195402 0.65 LTA4H (0.60) HRH3LTA4HLMNACYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1328512-A2 CYCLYLAMINE SULFONAMIDES AS BETA-3 ADRENERGIC RECEPTOR AGONISTS Wyeth (US) 2003-07-23 EP disclosed
WO-2002006221-A2 CYCLYLAMINE SULFONAMIDES AS BETA-3 ADRENERGIC RECEPTOR AGONISTS WYETH (US) 2002-01-24 WO disclosed