SCHEMBL6987673

SCHEMBL6987673

COc1ccc(C(=O)c2cccc(NCC(=O)NCC3CCN(C(C)C)CC3)c2Oc2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.43
ACHE P22303 1/20 0.43
ROCK2 O75116 2/20 0.41
HTR4 Q13639 2/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38
HRH3 Q9Y5N1 3/20 0.38
F10 P00742 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
MCL1 Q07820 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6984942 0.93 ROCK2 (0.42) FAAHACHEROCK2HTR4MEN1
SCHEMBL6986867 0.91 ROCK2 (0.41) FAAHACHEROCK2HTR4MEN1
SCHEMBL6988472 0.91 FAAH (0.46) FAAHACHEROCK2ALDH1A1SMN1; SMN2
SCHEMBL6983299 0.90 F10 (0.41) FAAHACHEROCK2HTR4MEN1
SCHEMBL6984041 0.89 ROCK2 (0.43) FAAHACHEROCK2HTR4MEN1
SCHEMBL6987182 0.88 FAAH (0.43) FAAHACHEROCK2HTR4MEN1
Hydrochloric Acid SCHEMBL6984317 0.87 ROCK2 (0.44) FAAHACHEROCK2HTR4MEN1
SCHEMBL6982360 0.87 HTR4 (0.42) FAAHACHEROCK2HTR4MEN1
SCHEMBL6989019 0.87 FAAH (0.42) FAAHACHEROCK2HTR4MEN1
SCHEMBL6985205 0.87 ROCK2 (0.42) FAAHACHEROCK2HTR4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289954-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096303-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed