SCHEMBL6987746

SCHEMBL6987746

CC(C)[Si](Oc1ccc(C(C=O)c2cccnc2)cc1)(C(C)C)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 2/20 0.37
KDM4E B2RXH2 2/20 0.35
CFTR P13569 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
GOPC Q9HD26 1/20 0.35
CYP19A1 P11511 3/20 0.35
MAPT P10636 1/20 0.34
ADRB3 P13945 2/20 0.34
CYP17A1 P05093 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6988582 0.84 CYP17A1 (0.35) KDM4ECYP19A1CYP17A1SMN1; SMN2LMNA
SCHEMBL6498908 0.83 KMT2A (0.46) KDM4ECYP19A1SMN1; SMN2
SCHEMBL6505294 0.78 ALDH1A1 (0.42) TBXAS1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL360712 0.77 CFTR (0.57) TBXAS1KDM4ECFTRSLC6A2SLC6A4
SCHEMBL6509102 0.77 ADRB3 (0.38) CYP19A1MAPTADRB3SMN1; SMN2LMNA
SCHEMBL6503338 0.75 CYP19A1 (0.62) CFTRSLC6A2SLC6A4SLC6A3GOPC
SCHEMBL6502611 0.75 POLB (0.51) CFTRSLC6A2SLC6A4SLC6A3GOPC
SCHEMBL6498870 0.74 ALDH1A1 (0.49) TBXAS1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL7492214 0.74 MAPK1 (0.54)
SCHEMBL8191216 0.73 PTGS2 (0.48) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1333827-A2 ESTROGEN RECEPTOR MODULATORS Merck & Co., Inc. (US) 2003-08-13 EP disclosed
EP-1328522-A2 ESTROGEN RECEPTOR MODULATORS Merck & Co., Inc. (US) 2003-07-23 EP disclosed
WO-2002032377-A2 ESTROGEN RECEPTOR MODULATORS MERCK & CO., INC. (US) 2002-04-25 WO disclosed
WO-2002032373-A2 ESTROGEN RECEPTOR MODULATORS MERCK & CO., INC. (US) 2002-04-25 WO disclosed