SCHEMBL6988076

SCHEMBL6988076

COC(=O)n1c(C(=O)O)cc2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.58
DAO P14920 1/20 0.56
ALDH1A1 P00352 3/20 0.53
TSHR P16473 1/20 0.53
CCR2 P41597 4/20 0.49
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
NOD2 Q9HC29 1/20 0.43
NOD1 Q9Y239 1/20 0.43
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
LDHA P00338 1/20 0.42
PHGDH O43175 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6988070 0.87 MTNR1A (0.51) MCL1DAOALDH1A1TSHRL3MBTL1
SCHEMBL7902953 0.83 NR1H2 (0.55) MCL1DAOALDH1A1TSHR
SCHEMBL29781083 0.83 NR1H2 (0.55) MCL1DAOALDH1A1TSHR
SCHEMBL4222282 0.81 MCL1 (0.64) MCL1DAOALDH1A1TSHRCCR2
SCHEMBL29780995 0.81 DAO (0.65) MCL1DAOALDH1A1TSHRCCR2
SCHEMBL3638561 0.81 DAO (0.65) MCL1DAOALDH1A1TSHRCCR2
SCHEMBL20909818 0.80 MCL1 (0.50) MCL1DAOALDH1A1TSHRL3MBTL1
SCHEMBL3831363 0.79 KDM1A (0.56) MCL1DAOALDH1A1TSHRCCR2
SCHEMBL14398966 0.79 MCL1 (0.60) MCL1DAOALDH1A1TSHRCCR2
SCHEMBL17075022 0.79 L3MBTL1 (0.47) MCL1DAOALDH1A1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1335917-A2 CONDENSED PYRIDOINDOLE DERIVATIVES Lilly Icos LLC (US) 2003-08-20 EP claimed
WO-2002028859-A2 CONDENSED PYRIDOINDOLE DERIVATIVES LILLY ICOS LLC (US) 2002-04-11 WO claimed