SCHEMBL6988745

SCHEMBL6988745

CC(C)c1ccc(C(=O)NCC(C(=O)NC23CCCC2OCC3=O)c2ccc(O)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.35
RAB9A P51151 5/20 0.35
SMN1; SMN2 Q16637 5/20 0.35
NPC1 O15118 4/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
DEGS1 O15121 1/20 0.34
ESRRG P62508 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
ALDH1A1 P00352 1/20 0.31
POLB P06746 2/20 0.31
MAPT P10636 1/20 0.31
TACR2 P21452 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994067 0.93 RAB9A (0.41) CTSKRAB9ASMN1; SMN2NPC1MEN1
SCHEMBL6294364 0.91 TP53 (0.38) CTSKRAB9AESRRGLMNAHPGD
SCHEMBL6993081 0.91 CTSK (0.35) CTSKRAB9ASMN1; SMN2NPC1MEN1
SCHEMBL6989694 0.91 KMT2A (0.40) SMN1; SMN2NPC1MEN1KMT2ALMNA
SCHEMBL6997966 0.90 MEN1 (0.34) MEN1KMT2ADEGS1OPRM1OPRD1
SCHEMBL6992764 0.89 HPGD (0.39) CTSKRAB9ASMN1; SMN2NPC1MEN1
SCHEMBL6993342 0.88 KMT2A (0.40) RAB9ASMN1; SMN2NPC1MEN1KMT2A
SCHEMBL6998484 0.87 TRPV1 (0.39)
SCHEMBL6989614 0.85 TP53 (0.47) CTSKRAB9ASMN1; SMN2NPC1MEN1
SCHEMBL6988021 0.85 NPC1 (0.39) SMN1; SMN2NPC1KMT2ALMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358176-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-05 EP disclosed
WO-2002057246-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed