SCHEMBL6992764

SCHEMBL6992764

CC(C)c1ccc(C(=O)NCC(C(=O)NC23CCCC2OCC3=O)c2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.39
SLC6A3 Q01959 5/20 0.35
GLP1R P43220 1/20 0.34
GCGR P47871 1/20 0.34
CTSK P43235 1/20 0.34
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
NPC1 O15118 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
TAOK1 Q7L7X3 1/20 0.33
TAOK3 Q9H2K8 1/20 0.33
KDM4E B2RXH2 1/20 0.33
KCNQ2 O43526 1/20 0.33
NFE2L2 Q16236 1/20 0.33
AKT1 P31749 1/20 0.32
CCR3 P51677 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996937 0.93 TP53 (0.40) HPGDSLC6A3GLP1RGCGRCTSK
SCHEMBL6986470 0.92 HPGD (0.38) HPGDSLC6A3GLP1RGCGRSMN1; SMN2
SCHEMBL6992598 0.91 AKT1 (0.38) HPGDSLC6A3GLP1RGCGRMEN1
SCHEMBL6994067 0.91 RAB9A (0.41) CTSKRAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL6988745 0.89 CTSK (0.35) HPGDCTSKRAB9ASMN1; SMN2MEN1
SCHEMBL6993081 0.89 CTSK (0.35) CTSKRAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7144829 0.88 TRPV1 (0.42) GCGRPTGDR2TAOK1TAOK3CCR3
SCHEMBL6989614 0.83 TP53 (0.47) GCGRCTSKRAB9ASMN1; SMN2MEN1
SCHEMBL6988021 0.83 NPC1 (0.39) HPGDSMN1; SMN2KMT2ANPC1LMNA
SCHEMBL6702836 0.82 CTSL (0.41) CTSKTAOK1TAOK3CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358176-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-05 EP disclosed
WO-2002057246-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed