SCHEMBL6989160

SCHEMBL6989160

CC(C)(C)OC(=O)NCCOc1noc2c(Cl)cc(Cl)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
STK17B O94768 1/20 0.40
STK17A Q9UEE5 1/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
HTT P42858 2/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
TP53 P04637 1/20 0.39
GLA P06280 1/20 0.39
MAPT P10636 1/20 0.39
XBP1 P17861 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989360 0.90 IDO1 (0.39) IDO1STK17BSTK17AALDH1A1HPGD
SCHEMBL6987117 0.88 KCNH2 (0.39) IDO1STK17BSTK17AALDH1A1HPGD
SCHEMBL6987906 0.88 CA12 (0.40) IDO1STK17BSTK17AALDH1A1HPGD
SCHEMBL6986485 0.85 LMNA (0.44) IDO1STK17BSTK17AHPGDCA12
SCHEMBL6991027 0.83 STK17B (0.40) IDO1STK17BSTK17AALDH1A1HPGD
SCHEMBL6989587 0.83 FAAH (0.49) IDO1ALDH1A1HPGDHTTCA12
SCHEMBL6988466 0.82 STK17B (0.40) IDO1STK17BSTK17AALDH1A1HPGD
SCHEMBL6988016 0.80 ALDH1A1 (0.49) IDO1ALDH1A1HPGDHTTCA12
SCHEMBL6990326 0.80 CA12 (0.39) IDO1HTTCA12CA1CA2
SCHEMBL6995142 0.80 IDO1 (0.47) IDO1STK17BSTK17AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779281-B1 ISOXAZOLES SANKYO CO (JP) 2003-10-29 EP disclosed
US-6096771-A ISOXAZOLE DERIVATIVES EXHIBITING EXCELLENT TYPE B AND TYPE A MONOAMINE OXIDASE INHIBITORY ACTIVITIES, THEREFORE USEFUL FOR PREVENTING PARKINSON'S DISEASE, DEPRESSION AND ALZHEIMER'S DISEASE SANKYO COMPANY, LIMITED (JP) 2000-08-01 US disclosed
US-5965591-A MONOAMINE OXIDASE INHIBITOR; FOR PROPHYLAXIS AND TREATING PARKINSON'S DISEASE, DEPRESSION AND ALZHEIMER'S DISEASE SANKYO COMPANY, LIMITED (JP) 1999-10-12 US disclosed
EP-0779281-A1 ISOXAZOLES SANKYO COMPANY LIMITED (JP) 1997-06-18 EP disclosed