SCHEMBL6989241

SCHEMBL6989241

COc1c(C)ccc2onc(OCCN)c12

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.33
MGLL Q99685 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989173 0.84 FAAH (0.35) FAAHMGLL
SCHEMBL6996361 0.83 FAAH (0.35) FAAHMGLL
Hydrochloric Acid SCHEMBL6988527 0.83 FAAH (0.35) FAAHMGLL
SCHEMBL8201516 0.82 FAAH (0.34) FAAHMGLL
Hydrochloric Acid SCHEMBL6989236 0.81 FAAH (0.33) FAAHMGLL
Hydrochloric Acid SCHEMBL6993053 0.80 KDM4E (0.33) FAAHMGLL
SCHEMBL6989250 0.80 FAAH (0.33) FAAHMGLL
SCHEMBL6997384 0.78 LMNA (0.32) FAAHMGLL
SCHEMBL6989881 0.78 FAAH (0.41) FAAHMGLL
SCHEMBL6988537 0.78 ALDH1A1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779281-B1 ISOXAZOLES SANKYO CO (JP) 2003-10-29 EP claimed
EP-0779281-A1 ISOXAZOLES SANKYO COMPANY LIMITED (JP) 1997-06-18 EP claimed
EP-0779281-B1 ISOXAZOLES SANKYO CO (JP) 2003-10-29 EP disclosed
US-6096771-A ISOXAZOLE DERIVATIVES EXHIBITING EXCELLENT TYPE B AND TYPE A MONOAMINE OXIDASE INHIBITORY ACTIVITIES, THEREFORE USEFUL FOR PREVENTING PARKINSON'S DISEASE, DEPRESSION AND ALZHEIMER'S DISEASE SANKYO COMPANY, LIMITED (JP) 2000-08-01 US disclosed
US-5965591-A MONOAMINE OXIDASE INHIBITOR; FOR PROPHYLAXIS AND TREATING PARKINSON'S DISEASE, DEPRESSION AND ALZHEIMER'S DISEASE SANKYO COMPANY, LIMITED (JP) 1999-10-12 US disclosed
EP-0779281-A1 ISOXAZOLES SANKYO COMPANY LIMITED (JP) 1997-06-18 EP disclosed