SCHEMBL6989374

SCHEMBL6989374

NC(=O)CCc1cccc(C(N)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.50
MEP1B Q16820 1/20 0.49
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
FOLH1 Q04609 1/20 0.46
CAPN1 P07384 1/20 0.44
IDH1 O75874 1/20 0.44
F10 P00742 3/20 0.44
F2 P00734 1/20 0.44
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
KDM1A O60341 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
TSHR P16473 2/20 0.43
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11119221 0.87 KEAP1 (0.57) PARP1MEP1BFOLH1TSHRPOLB
SCHEMBL1405064 0.86 ALDH1A1 (0.56) PARP1MEP1BMEN1KMT2AFOLH1
SCHEMBL8415332 0.84 L3MBTL1 (0.47) PARP1MEP1BMEN1KMT2AFOLH1
SCHEMBL10189495 0.83 PARP1 (0.56) PARP1MEP1BFOLH1KDM1AMAOA
SCHEMBL3054119 0.83 CYP4F2 (0.62) PARP1MEP1BFOLH1IDH1F10
SCHEMBL8342426 0.83 TAAR1 (0.55) PARP1MEP1BFOLH1
SCHEMBL23582699 0.82 CYP4F2 (0.69) PARP1MEN1KMT2AFOLH1CYP4F2
SCHEMBL5232156 0.81 PARP1 (0.53) PARP1MEP1BFOLH1IDH1F10
SCHEMBL5645749 0.81 PARP1 (0.53) PARP1MEP1BFOLH1IDH1F10
Hydrochloric Acid SCHEMBL28744996 0.81 TAAR1 (0.53) PARP1MEP1BFOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1341755-A1 CARBOXYLIC ACID AMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF THROMBOEMBOLIC DISEASES AND TUMOURS MERCK PATENT GmbH (DE) 2003-09-10 EP claimed
WO-2002048099-A1 CARBOXYLIC ACID AMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF THROMBOEMBOLIC DISEASES AND TUMOURS MERCK PATENT GMBH (DE) 2002-06-20 WO claimed