SCHEMBL6989880

SCHEMBL6989880

CC(C)(C)OC(=O)NC(=N)c1cc2c(s1)CC(C(=O)O)CC2

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 3/20 0.39
ALDH1A1 P00352 6/20 0.36
HPGD P15428 2/20 0.36
TP53 P04637 1/20 0.36
MAPK1 P28482 1/20 0.36
BTK Q06187 1/20 0.36
NPC1 O15118 2/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
KMT2A Q03164 2/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
PDK1 Q15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974020 0.86 ALDH1A1 (0.32) ALDH1A1HPGDTP53MAPK1NPC1
SCHEMBL7973903 0.84 ALDH1A1 (0.36) ALDH1A1HPGDTP53MAPK1NPC1
Hydrochloric Acid SCHEMBL6990489 0.74 TBXAS1 (0.46) TBXAS1ALDH1A1HPGDTP53MAPK1
SCHEMBL9871883 0.68 TBXAS1 (0.51) TBXAS1ALDH1A1NPC1RAB9APDK1
SCHEMBL31563842 0.65 EPHX2 (0.44) ALDH1A1HPGDMAPK1BTKNPC1
SCHEMBL31564285 0.65 EPHX2 (0.41) BTKKMT2AL3MBTL1
SCHEMBL31563886 0.64 ALDH1A1 (0.43) TBXAS1ALDH1A1HPGDTP53MAPK1
Hydrochloric Acid SCHEMBL6998122 0.64 PDK1 (0.47) ALDH1A1HPGDMAPK1NPC1POLB
SCHEMBL1397675 0.64 ALDH1A1 (0.53) ALDH1A1HPGDTP53MAPK1NPC1
Hydrochloric Acid SCHEMBL6998111 0.64 PDK1 (0.46) ALDH1A1HPGDMAPK1NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927177-B1 NOVEL BENZOTHIOPHENE DERIVATIVES, THEIR PREPARATION AND USE AS UROKINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO (JP) 2003-11-26 EP disclosed
US-6274619-B1 FUSED AMIDINO TYPE COMPOUNDS SUCH AS 4-(N-BUTYLCARBAMOYLMETHYLIDENE)-2-AMIDINO-4,5,6,7-TETRAHYDROBE NZO(B)THIOPHENE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-08-14 US disclosed