SCHEMBL6990108

SCHEMBL6990108

COc1cc(C(=CC=O)c2cc(-c3cccs3)ccc2OC)ccc1O

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 12/20 0.60
ERN1 O75460 3/20 0.46
ABCB1 P08183 1/20 0.44
ABCC1 P33527 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986840 0.83 TNFRSF1A (0.65) TNFRSF1AKDM4EALDH1A1
SCHEMBL4628631 0.78 TNFRSF1A (0.60) TNFRSF1AERN1MEN1KMT2AKDM4E
SCHEMBL7062708 0.77 TNFRSF1A (0.50) TNFRSF1AERN1MEN1KMT2AKDM4E
SCHEMBL6988312 0.76 TNFRSF1A (0.44) TNFRSF1AERN1
SCHEMBL7121640 0.76 TNFRSF1A (0.64) TNFRSF1AHDAC1HDAC2RAB9A
SCHEMBL5575668 0.75 TNFRSF1A (1.00) TNFRSF1A
SCHEMBL5575661 0.75 TNFRSF1A (1.00) TNFRSF1A
SCHEMBL6985223 0.75 ERN1 (0.49) TNFRSF1AERN1ABCB1ABCC1MEN1
SCHEMBL6990105 0.74 TNFRSF1A (0.60) TNFRSF1AERN1KDM4EL3MBTL1RAB9A
SCHEMBL6093064 0.73 TNFRSF1A (0.52) TNFRSF1AABCB1ABCC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1330448-A2 1,3-BIS-(SUBSTITUTED-PHENYL)-2-PROPEN-1-ONES AND THEIR USE TO TREAT VCAM-1 MEDIATED DISORDERS Atherogenics, Inc. (US) 2003-07-30 EP claimed
WO-2001098291-A2 1,3-BIS-(SUBSTITUTED-PHENYL)-2-PROPEN-1-ONES AND THEIR USE TO TREAT VCAM-1 MEDIATED DISORDERS ATHEROGENICS, INC. (US) 2001-12-27 WO claimed