SCHEMBL6990562

SCHEMBL6990562

CC(C)(C)OC(=O)C(C1CCNCC1)N1CCN(C(=O)CN(C(=O)OCc2ccccc2)c2ccccc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 2/20 0.40
CACNA1B Q00975 2/20 0.40
CACNB1 Q02641 2/20 0.40
CTSL P07711 1/20 0.39
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
MAPT P10636 2/20 0.34
CCR5 P51681 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPK1 P28482 1/20 0.34
NTSR1 P30989 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
FKBP1A P62942 1/20 0.34
ALDH1A1 P00352 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985406 0.83 ACHE (0.44) CACNA2D1CACNA1BCACNB1MAPTMEN1
SCHEMBL4842101 0.80 MEN1 (0.46) CHRM2CHRM1CHRM3MAPTMEN1
SCHEMBL4832645 0.79 CHRM2 (0.44) CACNA2D1CACNA1BCACNB1CHRM2CHRM5
SCHEMBL6989033 0.77 CACNA2D1 (0.45) CACNA2D1CACNA1BCACNB1SIGMAR1MEN1
SCHEMBL4838599 0.75 KDM4E (0.44) CACNA2D1CACNA1BCACNB1CHRM2CHRM1
SCHEMBL6580060 0.74 KCNA3 (0.47) CTSLMAPTCCR5MEN1KMT2A
SCHEMBL6369665 0.74 ALDH1A1 (0.47) CHRM2CHRM5CHRM1CHRM3SIGMAR1
SCHEMBL4385892 0.73 SMN1; SMN2 (0.42) CTSLSIGMAR1MEN1KMT2ANPSR1
SCHEMBL4840733 0.72 KDM4E (0.46) CHRM2CHRM5CHRM1CHRM3SIGMAR1
SCHEMBL5868123 0.72 ITGB3 (0.40) ITGB3ITGA2BCHRM2CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289972-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096323-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed