SCHEMBL6991969

SCHEMBL6991969

Cc1c(CO)c2cccc(Cl)c2[nH]c1=O

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
DAO P14920 2/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HPGD P15428 2/20 0.42
KDM4E B2RXH2 2/20 0.42
RXFP1 Q9HBX9 1/20 0.41
TSHR P16473 2/20 0.41
PARP1 P09874 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
MAP2 P11137 1/20 0.40
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
AR P10275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998461 0.81 KDM4E (0.49) L3MBTL1DAOMEN1KMT2AHPGD
SCHEMBL3641835 0.80 DAO (0.49) DYRK1AL3MBTL1DAOMEN1KMT2A
SCHEMBL20669916 0.76 DAO (0.59) DAOMEN1KMT2AHPGDKDM4E
SCHEMBL19846959 0.72 DYRK1A (0.55) DYRK1AL3MBTL1MEN1KMT2AHPGD
SCHEMBL29432610 0.72 DYRK1A (0.55) DYRK1AL3MBTL1MEN1KMT2AHPGD
SCHEMBL6991966 0.70 MEN1 (0.52) DYRK1AMEN1KMT2AHPGDKDM4E
SCHEMBL18509923 0.69 L3MBTL1 (0.46) DYRK1AL3MBTL1MEN1KMT2AHPGD
SCHEMBL3383227 0.69 MAPT (0.55) DYRK1AL3MBTL1MEN1KMT2AHPGD
SCHEMBL14566728 0.68 DAO (0.53) DYRK1ADAOKDM4EPARP1MAP2
SCHEMBL4076852 0.68 KDM4E (0.62) DYRK1AL3MBTL1MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003724-B1 SUBSTITUTED QUINOLINE DERIVATIVES WITH ANTIVIRAL ACTION AVENTIS PHARMA GMBH (DE) 2003-02-12 EP disclosed