SCHEMBL6992847

SCHEMBL6992847

CCCCC1(CC)C(=O)Sc2cc(OCC(=O)OCC)c(SC)cc2N(c2ccccc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ELANE P08246 3/20 0.43
CYP2C19 P33261 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
PKM P14618 2/20 0.34
KDM4E B2RXH2 2/20 0.34
NR1H4 Q96RI1 1/20 0.33
ABCB1 P08183 1/20 0.33
CASP3 P42574 1/20 0.33
CASP7 P55210 1/20 0.33
CASP9 P55211 1/20 0.33
GAA P10253 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
PPOX P50336 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
ATM Q13315 1/20 0.32
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7507444 0.90 ELANE (0.45) ELANECYP2C19NPC1RAB9APKM
SCHEMBL6986488 0.89 GAA (0.36) ELANENPC1RAB9APKMKDM4E
SCHEMBL6993818 0.88 ELANE (0.43) ELANECYP2C19PKMKDM4ENR1H4
SCHEMBL6993226 0.88 ELANE (0.41) ELANECYP2C19PKMKDM4EALDH1A1
SCHEMBL6993400 0.87 ELANE (0.42) ELANECYP2C19NPC1RAB9APKM
SCHEMBL6993131 0.85 ELANE (0.41) ELANECYP2C19NPC1RAB9APKM
SCHEMBL7513280 0.82 ELANE (0.44) ELANECYP2C19PKMKDM4EGAA
SCHEMBL6994314 0.82 ELANE (0.52) ELANECYP2C19PKMKDM4EALDH1A1
Ethyl Bromo Acetate SCHEMBL7509727 0.82 ALDH1A1 (0.39) ELANECYP2C19NPC1RAB9APKM
SCHEMBL3835251 0.81 NR1H4 (0.44) ELANEKDM4ENR1H4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1345918-A1 CHEMICAL COMPOUNDS AstraZeneca AB (SE) 2003-09-24 EP disclosed
EP-1263747-A1 1,5-BENZOTHIAZEPINES AND THEIR USE AS HYPOLIPIDAEMICS AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2002050051-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2002-06-27 WO disclosed
WO-2001066533-A1 1,5-BENZOTHIAZEPINES AND THEIR USE AS HYPOLIPIDAEMICS ASTRAZENECA AB (SE) 2001-09-13 WO disclosed