SCHEMBL6993873

SCHEMBL6993873

O=C(O)NS(=O)(=O)NCc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.70
CA2 P00918 4/20 0.70
CA7 P43166 3/20 0.70
CA14 Q9ULX7 3/20 0.70
CA1 P00915 4/20 0.67
KEAP1 Q14145 1/20 0.53
LMNA P02545 2/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 1/20 0.53
CA9 Q16790 2/20 0.51
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 1/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TSHR P16473 2/20 0.47
MEN1 O00255 1/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
RECQL P46063 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14798746 0.84 CA2 (0.49) CA12CA2CA7CA14CA1
SCHEMBL3194925 0.84 SMN1; SMN2 (0.54) CA12CA2CA7CA14CA1
Benzyl(Benzylsulfamoyl)Amine SCHEMBL2298224 0.83 CA12 (1.00) CA12CA2CA7CA14CA1
SCHEMBL12002489 0.83 CA2 (0.49) CA12CA2CA7CA14CA1
SCHEMBL30136175 0.82 CA12 (0.68) CA12CA2CA7CA14CA1
SCHEMBL3209241 0.81 CA12 (0.60) CA12CA7CA14LMNAKMT2A
SCHEMBL3211224 0.80 HTT (0.69) CA12CA7CA14CA1LMNA
SCHEMBL6337412 0.77 CA12 (1.00) CA12CA2CA7CA14CA1
SCHEMBL3195623 0.76 L3MBTL1 (0.56) KMT2AATML3MBTL1MEN1KDM4E
SCHEMBL1134868 0.76 CA2 (0.76) CA12CA2CA7CA14CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874809-B1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-08-27 EP claimed
US-6239175-B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-29 US claimed
US-11850286-B2 Sulfamide linker, conjugates thereof, and methods of preparation SYNAFFIX B.V. (NL) 2023-12-26 US disclosed
US-20210030886-A1 SULFAMIDE LINKER, CONJUGATES THEREOF, AND METHODS OF PREPARATION SYNAFFIX B.V. (NL) 2021-02-04 US disclosed
US-10792369-B2 Sulfamide linker, conjugates thereof, and methods of preparation SYNAFFIX B.V. (NL) 2020-10-06 US disclosed
US-20170298145-A1 SULFAMIDE LINKER, CONJUGATES THEREOF, AND METHODS OF PREPARATION SYNAFFIX B.V. (NL) 2017-10-19 US disclosed
US-9636421-B2 Sulfamide linker, conjugates thereof, and methods of preparation SYNAFFIX B.V. (NL) 2017-05-02 US disclosed
EP-0874809-B1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-08-27 EP disclosed
US-6239175-B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-29 US disclosed
US-6020368-A MICROBIOCIDES HINKS JEREMY DAVID (US) 2000-02-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170298145-A1 SULFAMIDE LINKER, CONJUGATES THEREOF, AND METHODS OF PREPARATION SULT1E1, SULT1A1, SULT2A1 CA12 654/4885CA2 1487/4885CA7 1918/4885
US-10792369-B2 Sulfamide linker, conjugates thereof, and methods of preparation SULT1E1, SULT1A1, SULT2A1 CA12 654/4885CA2 1487/4885CA7 1918/4885
US-11850286-B2 Sulfamide linker, conjugates thereof, and methods of preparation SULT1E1, SULT1A1, SULT2A1 CA12 654/4885CA2 1487/4885CA7 1918/4885
US-20210030886-A1 SULFAMIDE LINKER, CONJUGATES THEREOF, AND METHODS OF PREPARATION SULT1E1, SULT1A1, SULT2A1 CA12 654/4885CA2 1487/4885CA7 1918/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.