SCHEMBL6994359

SCHEMBL6994359

COC(=O)c1cccc(N2CCN(c3ccc(-c4nc5cc(Cl)ccc5[nH]4)cn3)CC2)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.50
DGAT1 O75907 11/20 0.49
KCNH2 Q12809 6/20 0.49
ADORA2A P29274 2/20 0.49
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45
RHEB Q15382 1/20 0.45
CYP2C9 P11712 1/20 0.43
MCL1 Q07820 1/20 0.43
MGLL Q99685 1/20 0.43
DGAT2 Q96PD7 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993769 0.90 CHEK2 (0.53) CHEK2DGAT1KCNH2ADORA2ADRD2
SCHEMBL1687861 0.86 RET (0.47) DGAT1KCNH2ADORA2AMGLLDGAT2
SCHEMBL14235564 0.84 DGAT1 (0.53) CHEK2DGAT1KCNH2ADORA2ADGAT2
SCHEMBL6994712 0.82 DGAT1 (0.54) CHEK2DGAT1KCNH2ADORA2AKMT2A
SCHEMBL4559775 0.82 DGAT1 (0.49) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL10081696 0.81 DGAT1 (0.48) DGAT1KCNH2ADORA2ANPC1RAB9A
SCHEMBL4543375 0.81 CHEK2 (0.59) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL4561622 0.80 DGAT1 (0.48) CHEK2DGAT1KCNH2ADORA2ADRD2
SCHEMBL4560992 0.80 DGAT1 (0.57) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL14128676 0.80 DGAT1 (0.55) CHEK2DGAT1KCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed