SCHEMBL10326124

SCHEMBL10326124

FC(F)(F)c1ccc2[nH]c(-c3ccc(-c4ccc(N5CCNCC5)nc4)cc3)nc2c1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 16/20 0.68
KCNH2 Q12809 7/20 0.68
SOAT1 P35610 4/20 0.68
PRMT5 O14744 1/20 0.53
ADORA2A P29274 2/20 0.53
NPBWR1 P48145 1/20 0.53
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4560514 0.96 DGAT1 (0.62) DGAT1KCNH2SOAT1PRMT5ADORA2A
SCHEMBL10381569 0.84 DGAT1 (0.62) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL10380785 0.84 DGAT1 (0.73) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL4561861 0.82 DGAT1 (0.65) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL1742865 0.82 GPR119 (0.57) DGAT1KCNH2SOAT1PRMT5
SCHEMBL10325481 0.81 DGAT1 (0.62) DGAT1KCNH2SOAT1PRMT5ADORA2A
SCHEMBL19175769 0.81 DGAT1 (0.77) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL4566517 0.80 DGAT1 (0.60) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL6995535 0.80 DGAT1 (0.61) DGAT1KCNH2SOAT1ADORA2ACYP3A4
SCHEMBL1687841 0.79 HTR3E (0.54) DGAT1KCNH2SOAT1ADORA2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096813-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-07-19 WO disclosed