SCHEMBL6995912

SCHEMBL6995912

Cc1csc(-c2[nH]c(-c3ccccc3)c3c2CC=CC3)c1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.34
KDR P35968 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 2/20 0.31
HPGD P15428 1/20 0.31
HPGDS O60760 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990226 0.86 BRD4 (0.43) BRD4KDRSMN1; SMN2KDM4E
SCHEMBL6998152 0.78 KDM4E (0.44) BRD4KDM4EHPGDALDH1A1GAA
SCHEMBL72613 0.72 AR (0.43) SMN1; SMN2HPGDCYP3A4CYP2C19
SCHEMBL6998491 0.72 KDR (0.35) BRD4KDRKDM4EHPGDALDH1A1
SCHEMBL6995905 0.68 PTGS2 (0.46) KDM4EHPGDMEN1ALDH1A1CYP1A2
SCHEMBL7093334 0.68 KDM4E (0.46) SMN1; SMN2KDM4EHPGDALDH1A1GAA
SCHEMBL7567903 0.67 PTGS2 (0.34) SMN1; SMN2HPGDHPGDS
SCHEMBL10892833 0.67 KDM4E (0.56) KDM4ECYP3A4
SCHEMBL7093332 0.66 HSD17B10 (0.44) SMN1; SMN2KDM4EHPGDALDH1A1CYP1A2
SCHEMBL10472855 0.65 HSD17B1 (0.47) SMN1; SMN2KDM4EHPGDMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0921119-B1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-07-02 EP disclosed
US-6114360-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-09-05 US disclosed
US-6063804-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-05-16 US disclosed
EP-0921119-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-06-09 EP disclosed