SCHEMBL6995905

SCHEMBL6995905

CSc1ccc(-c2[nH]c(-c3ccccc3)c3c2CC=CC3)cc1

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.46
GSK3B P49841 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGS1 P23219 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
ALDH1A3 P47895 1/20 0.36
NISCH Q9Y2I1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998152 0.84 KDM4E (0.44) KDM4EALDH1A1HPGDGAA
SCHEMBL6990217 0.83 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL6998482 0.75 CDKN1A (0.44) PTGS2KDM4EHPGDPTGS1NISCH
SCHEMBL403028 0.73 PTGS2 (0.63) PTGS2GSK3BALDH1A1PTGS1MEN1
SCHEMBL17283465 0.73 PTGS2 (0.63) PTGS2GSK3BALDH1A1PTGS1MEN1
Hydrogen Sulfide SCHEMBL19086306 0.71 PTGS2 (0.61) PTGS2GSK3BALDH1A1PTGS1MEN1
SCHEMBL7567894 0.69 PTGS2 (0.53) PTGS2GSK3BKDM4EALDH1A1HPGD
SCHEMBL29158890 0.68 PTGS2 (0.41) PTGS2GSK3BKDM4EMEN1KMT2A
SCHEMBL6995912 0.68 BRD4 (0.34) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL1131081 0.68 MAPK13 (0.67) GSK3BKDM4EALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0921119-B1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-07-02 EP disclosed
US-6114360-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-09-05 US disclosed
US-6063804-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-05-16 US disclosed
EP-0921119-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-06-09 EP disclosed