SCHEMBL6996474

SCHEMBL6996474

N#Cc1ccc2c(ccn2CC2CCN(Cc3cccc(Cl)c3)C2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CXCR4 P61073 1/20 0.40
P2RX7 Q99572 1/20 0.39
PRMT5 O14744 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CLPP Q16740 1/20 0.39
POLB P06746 1/20 0.39
DHFR P00374 1/20 0.39
CCR3 P51677 1/20 0.38
ROCK2 O75116 2/20 0.38
CCR2 P41597 2/20 0.38
ACHE P22303 1/20 0.38
ROCK1 Q13464 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7945151 0.99 KDM4E (0.45) KDM4EALDH1A1GLAGAAMAPT
SCHEMBL6995870 0.93 KDM4E (0.47) KDM4EALDH1A1GLAGAAMAPT
Hydrochloric Acid SCHEMBL7954259 0.92 KDM4E (0.46) KDM4EALDH1A1GLAGAAMAPT
SCHEMBL6991633 0.91 P2RX7 (0.47) P2RX7PRMT5CCR3ACHE
Hydrochloric Acid SCHEMBL7950551 0.90 P2RX7 (0.46) P2RX7PRMT5ACHE
SCHEMBL6993372 0.84 ALDH1A1 (0.48) KDM4EALDH1A1GLAHTTPRMT5
SCHEMBL6998552 0.84 HRH3 (0.43) KDM4EALDH1A1GLAGAAMAPT
SCHEMBL6997268 0.83 CXCR4 (0.45) ALDH1A1ATMCXCR4P2RX7PRMT5
Hydrochloric Acid SCHEMBL7950618 0.83 HRH3 (0.42) KDM4EALDH1A1GLAGAAMAPT
Hydrochloric Acid SCHEMBL7950497 0.83 ALDH1A1 (0.47) KDM4EALDH1A1GLAHTTPRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023898-B1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands SERVIER LAB (FR) 2003-03-12 EP disclosed
EP-1023898-A1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands ADIR ET COMPAGNIE (FR) 2000-08-02 EP disclosed