SCHEMBL6996665

SCHEMBL6996665

CC1=C(N)Nc2cc(CNCc3ccc(Cl)cc3Cl)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.39
POLB P06746 2/20 0.36
PARP1 P09874 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
LMNA P02545 2/20 0.35
MAPK1 P28482 1/20 0.35
NLRP1 Q9C000 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
GAA P10253 1/20 0.34
CYP2C19 P33261 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6998295 0.99 HTT (0.41) HTTPOLBPARP1MEN1KMT2A
SCHEMBL6993345 0.88 PARP1 (0.42) HTTPOLBPARP1MEN1KMT2A
Hydrochloric Acid SCHEMBL6996685 0.87 PARP1 (0.41) HTTPOLBPARP1MEN1KMT2A
Hydrochloric Acid SCHEMBL6998857 0.87 MEN1 (0.44) HTTPOLBPARP1MEN1KMT2A
SCHEMBL7002470 0.85 PARP1 (0.42) PARP1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL6993016 0.85 L3MBTL1 (0.45) POLBPARP1SMN1; SMN2CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL6996848 0.84 PARP1 (0.41) PARP1LMNACYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL6990749 0.84 L3MBTL1 (0.44) POLBPARP1MEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL6999676 0.80 PARP1 (0.43) POLBPARP1MEN1KMT2ATP53
Hydrochloric Acid SCHEMBL7000763 0.80 PARP1 (0.43) HTTPOLBPARP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP claimed