SCHEMBL6997020

SCHEMBL6997020

CC1=C(N)Nc2cc(C=CC#N)ccc2O1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.41
KDM4E B2RXH2 1/20 0.36
FDPS P14324 1/20 0.35
ENPP2 Q13822 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708170 1.00 ALOX5 (0.41) ALOX5KDM4EFDPSENPP2
SCHEMBL6992552 0.77 ALOX5 (0.49) ALOX5KDM4E
SCHEMBL7002017 0.76 ABL1 (0.35) KDM4E
SCHEMBL5670589 0.70 AHR (0.39)
SCHEMBL7711338 0.69 PARP1 (0.52) ALOX5KDM4EFDPS
SCHEMBL6994006 0.69 ALOX5 (0.36) ALOX5KDM4EFDPSENPP2
SCHEMBL6998554 0.69 PARP1 (0.52) ALOX5KDM4EFDPS
SCHEMBL5670592 0.69 ALOX5 (0.56) ALOX5
Hydrochloric Acid SCHEMBL5672533 0.69 AHR (0.38)
SCHEMBL7988325 0.68 ALDH1A1 (0.36) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP disclosed
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed