SCHEMBL6998079

SCHEMBL6998079

O=C(c1ccc(Br)cc1)C1CN(CCCc2ccccc2)CCC1(O)c1ccc(Br)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.64
ALDH1A1 P00352 4/20 0.64
LMNA P02545 3/20 0.64
MAPT P10636 3/20 0.62
MEN1 O00255 1/20 0.62
MAPK1 P28482 1/20 0.62
SLC6A3 Q01959 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
KCNH2 Q12809 1/20 0.46
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
HTR2A P28223 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002758 0.94 KMT2A (0.64) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL9710832 0.84 KMT2A (0.78) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL11743879 0.84 KMT2A (0.78) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL7003100 0.83 ALDH1A1 (0.53) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL6998218 0.82 SLC6A3 (0.64) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL9296977 0.81 KMT2A (0.69) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL11744954 0.79 KMT2A (0.81) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL13562203 0.78 KMT2A (1.00) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL11740905 0.78 KMT2A (1.00) KMT2AALDH1A1LMNAMAPTMEN1
SCHEMBL9714953 0.78 ALDH1A1 (0.83) KMT2AALDH1A1LMNAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP disclosed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP disclosed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO disclosed