SCHEMBL7003100

SCHEMBL7003100

O=C(c1ccccc1Br)C1CN(CCc2ccccc2)CCC1(O)c1ccc(Br)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
KMT2A Q03164 3/20 0.53
LMNA P02545 2/20 0.53
MAPT P10636 2/20 0.53
MEN1 O00255 1/20 0.53
MAPK1 P28482 1/20 0.53
OPRM1 P35372 9/20 0.42
ARRB1 P49407 1/20 0.42
OPRK1 P41145 6/20 0.39
OPRD1 P41143 4/20 0.39
HTR2A P28223 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
OPRL1 P41146 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002758 0.89 KMT2A (0.64) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL6998079 0.83 KMT2A (0.64) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL9710832 0.81 KMT2A (0.78) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL11743879 0.81 KMT2A (0.78) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL6995927 0.73 SLC6A3 (0.66) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL27563251 0.72 SIGMAR1 (0.68) OPRM1OPRK1OPRD1HTR2AOPRL1
SCHEMBL8967064 0.69 ALDH1A1 (1.00) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL11745258 0.69 KMT2A (0.77) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL8967060 0.69 ALDH1A1 (1.00) ALDH1A1KMT2ALMNAMAPTMEN1
SCHEMBL8967059 0.69 ALDH1A1 (1.00) ALDH1A1KMT2ALMNAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed