SCHEMBL6998427

SCHEMBL6998427

O=c1ccoc(CO)c1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.52
LMNA P02545 1/20 0.52
APP P05067 6/20 0.38
FTO Q9C0B1 2/20 0.37
TYR P14679 1/20 0.36
DAO P14920 1/20 0.36
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP12 P39900 1/20 0.36
MMP13 P45452 1/20 0.36
TEAD4 Q15561 1/20 0.35
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DBH P09172 2/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700110 0.83 KDM4E (0.48) KDM4ELMNAAPPFTOTYR
E637 SCHEMBL41817 0.81 KDM4E (0.55) KDM4ELMNAAPPFTOMMP1
E637 SCHEMBL1870685 0.81 KDM4E (0.55) KDM4ELMNAAPPFTOMMP1
SCHEMBL561713 0.81 KDM4E (0.50) KDM4ELMNAAPPFTOMMP1
E637 SCHEMBL8026696 0.79 KDM4E (0.53) KDM4ELMNAAPPFTOMMP1
E637 SCHEMBL27635951 0.79 KDM4E (0.53) KDM4ELMNAAPPFTOMMP1
E637 SCHEMBL6657728 0.79 KDM4E (0.53) KDM4ELMNAAPPFTOMMP1
SCHEMBL9625161 0.78 KDM4E (0.52) KDM4ELMNAAPPFTOMMP1
SCHEMBL9700079 0.78 KDM4E (0.47) KDM4ELMNAAPPFTOMMP1
SCHEMBL3316478 0.76 KDM4E (0.46) KDM4ELMNAAPPFTOMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109438405-B Synthetic method of 3- (benzyloxy) -4-oxo-4H-pyran-2-carboxylic acid 广东莱佛士制药技术有限公司 2023-04-07 CN claimed
CN-111320598-B Preparation method of hydroxypyrone compound 广东东阳光药业有限公司 2022-04-26 CN claimed
CN-111320598-A Preparation method of hydroxypyrone compound 广东东阳光药业有限公司 2020-06-23 CN claimed
JP-61197506-A None JP disclosed
CN-118702662-A Green technology for synthesizing 4-methyl-2H-pyran-2, 6 (3H) -dione 无锡小荷智化科技有限公司 2024-09-27 CN disclosed
CN-109438405-B Synthetic method of 3- (benzyloxy) -4-oxo-4H-pyran-2-carboxylic acid 广东莱佛士制药技术有限公司 2023-04-07 CN disclosed
CN-111320598-B Preparation method of hydroxypyrone compound 广东东阳光药业有限公司 2022-04-26 CN disclosed
CN-111320598-B Preparation method of hydroxypyrone compound 广东东阳光药业有限公司 2022-04-26 CN disclosed
CN-111606879-A Method for preparing 2-hydroxymethyl-3-alkoxy-4H-pyran-4-ketone by one-pot method 安徽金禾实业股份有限公司 2020-09-01 CN disclosed
WO-2020132820-A1 SYNTHESIS METHOD FOR 3-(BENZYLOXY)-4-OXO-4H-PYRAN-2-CARBOXYLIC ACID 广东莱佛士制药技术有限公司 2020-07-02 WO disclosed
WO-2020132820-A1 SYNTHESIS METHOD FOR 3-(BENZYLOXY)-4-OXO-4H-PYRAN-2-CARBOXYLIC ACID 广东莱佛士制药技术有限公司 2020-07-02 WO disclosed
US-20020068758-A1 Novel orally active iron (III) chelators BTG INTERNATIONAL LIMITED. 2002-06-06 US disclosed
US-6335353-B1 3-HYDROXYPYRIDIN-4-ONE DERIVATIVE; IRON DEFICIENCY ANEMIA AND THALASSEMIA TREATMENT BTG INTERNATIONAL LIMITED (GB) 2002-01-01 US disclosed
EP-0984934-A1 NOVEL ORALLY ACTIVE IRON (III) CHELATORS BTG INTERNATIONAL LIMITED (Company No. 2664412) (GB) 2000-03-15 EP disclosed
WO-1998054138-A1 NOVEL ORALLY ACTIVE IRON (III) CHELATORS BTG INTERNATIONAL LIMITED (GB) 1998-12-03 WO disclosed
WO-1992012131-A1 3-HYDROXYPYRIDIN-4-ONE DERIVATIVES AS PHARMACEUTICAL COMPOSITIONS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1992-07-23 WO disclosed
EP-0494754-A1 3-hydroxypyridin-4-one derivatives as pharmaceutical compositions BRITISH TECHNOLOGY GROUP LTD (GB) 1992-07-15 EP disclosed
JP-S61197506-A PREVENTION OF COLOR-BLACKENING OF LIVING BODIES WITH GAMMA-PYRONE DERIVATIVE YAKURIGAKU CHUO KENKYUSHO:KK 1986-09-01 JP disclosed
US-4219483-A 4-Pyrone prostaglandin antagonists PFIZER INC. (US) 1980-08-26 US disclosed
US-4132847-A 4-Pyrone prostaglandin antagonists PFIZER INC. (US) 1979-01-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020068758-A1 Novel orally active iron (III) chelators HAMP, HRH2, GRHPR KDM4E 1012/4885LMNA 2634/4885APP 4051/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.