SCHEMBL7001329

SCHEMBL7001329

CN1Cc2cccnc2C(=O)c2ccc(Cl)cc21

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
FNTA P49354 7/20 0.44
FNTB P49356 7/20 0.44
HRH1 P35367 4/20 0.42
PTAFR P25105 4/20 0.42
SLC6A15 Q9H2J7 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002677 0.75 LMNA (0.43) LMNASMN1; SMN2
SCHEMBL3839936 0.75 HRH1 (0.60) LMNAFNTAFNTBHRH1PTAFR
SCHEMBL29413038 0.75 HRH1 (0.60) LMNAFNTAFNTBHRH1PTAFR
SCHEMBL21971002 0.73 LMNA (0.46) LMNASMN1; SMN2FNTAFNTBHRH1
SCHEMBL6998860 0.72 FNTA (0.49) LMNAFNTAFNTBHRH1PTAFR
SCHEMBL6996504 0.71 FNTA (0.51) LMNAFNTAFNTBHRH1PTAFR
SCHEMBL29431445 0.71 ADAM17 (0.48) LMNASMN1; SMN2HRH1
SCHEMBL12573365 0.71 ADAM17 (0.48) LMNASMN1; SMN2HRH1
SCHEMBL6999299 0.70 FNTA (0.52) LMNAFNTAFNTBHRH1PTAFR
SCHEMBL6994178 0.69 FNTA (0.56) LMNASMN1; SMN2FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021448-B1 TRICYCLIC COMPOUNDS HAVING ACTIVITY AS Ras-FPT INHIBITORS SCHERING CORP (US) 2003-05-02 EP disclosed
US-6130229-A Tricyclic compounds having activity as RAS-FPT inhibitors SCHERING CORPORATION (US) 2000-10-10 US disclosed
EP-1021448-A1 TRICYCLIC COMPOUNDS HAVING ACTIVITY AS Ras-FPT INHIBITORS SCHERING CORPORATION (US) 2000-07-26 EP disclosed
WO-1998015556-A1 TRICYCLIC COMPOUNDS HAVING ACTIVITY AS Ras-FPT INHIBITORS SCHERING CORPORATION (US) 1998-04-16 WO disclosed