SCHEMBL7001987

SCHEMBL7001987

Cc1ccc(C(=O)C2CNCCC2(CO)c2ccc(C)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.43
MEN1 O00255 2/20 0.43
CYP2D6 P10635 2/20 0.43
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
GABRA4 P48169 1/20 0.39
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
SLC6A3 Q01959 2/20 0.33
OPRM1 P35372 1/20 0.33
HTT P42858 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001284 0.88 LMNA (0.44) KMT2AALDH1A1LMNAMAPTSLC6A3
SCHEMBL7001738 0.87 ALDH1A1 (0.36) KMT2APOLBALDH1A1LMNAMAPT
SCHEMBL7003750 0.87 LMNA (0.33) KMT2APOLBALDH1A1LMNAMAPT
SCHEMBL6995034 0.83 SLC6A3 (0.38) KMT2AMEN1CYP2D6ALDH1A1SLC6A3
SCHEMBL7002089 0.81 SLC6A2 (0.39) CYP2D6SLC6A3SLC6A2SLC6A4
SCHEMBL7004831 0.78 REN (0.42) SLC6A3SLC6A2SLC6A4
SCHEMBL7005083 0.73 SLC6A4 (0.41) SLC6A3SLC6A2SLC6A4
SCHEMBL7002761 0.71 LMNA (0.34) KMT2AMEN1POLBALDH1A1LMNA
SCHEMBL7003952 0.69 SLC6A4 (0.51) SLC6A3SLC6A2SLC6A4
SCHEMBL8967555 0.67 KMT2A (0.56) KMT2AMEN1ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP disclosed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP disclosed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO disclosed