SCHEMBL7002487

SCHEMBL7002487

N#Cc1c[nH]c2cc3c(cc2c1=O)OCCO3

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
RAB9A P51151 3/20 0.50
LMNA P02545 3/20 0.50
TP53 P04637 2/20 0.50
NPC1 O15118 2/20 0.44
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KDM4E B2RXH2 4/20 0.40
HTT P42858 2/20 0.40
HPGD P15428 2/20 0.40
IMPDH2 P12268 1/20 0.37
IMPDH1 P20839 1/20 0.37
XDH P47989 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
HASPIN Q8TF76 1/20 0.35
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL980263 0.78 HTR3E (0.48) ALDH1A1MAPTNPSR1KDM4EIMPDH2
SCHEMBL5329622 0.74 GPR84 (0.44) KDM4EIMPDH2IMPDH1CCNT1CDK9
SCHEMBL1200586 0.73 SMN1; SMN2 (0.71) ALDH1A1SMN1; SMN2RAB9ALMNATP53
SCHEMBL4992479 0.72 CCNT1 (0.52) ALDH1A1KDM4EHPGDIMPDH2IMPDH1
SCHEMBL4765036 0.71 KDM4E (0.47) ALDH1A1SMN1; SMN2LMNAMAPTKDM4E
SCHEMBL8320200 0.70 IMPDH2 (0.37) KDM4EIMPDH2IMPDH1XDHCCNT1
SCHEMBL27680529 0.70 GPR84 (0.50) ALDH1A1IMPDH2IMPDH1CCNT1CDK9
SCHEMBL5322018 0.69 IMPDH2 (0.46) ALDH1A1LMNAMAPTNPSR1KDM4E
SCHEMBL13202452 0.69 NR4A2 (0.44) ALDH1A1RAB9ATP53NPC1KDM4E
SCHEMBL3882080 0.69 IMPDH2 (0.46) IMPDH2IMPDH1XDHCCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117659-B1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS WYETH CORP (US) 2003-12-03 EP disclosed
US-6288082-B1 COMPOUNDS SUCH AS 6,7-DIETHOXY-4-(INDAN-5-YLAMINO) -QUINOLINE-3-CARBONITRILE USED AS ANTINEOPLASTIC AGENTS AND IN THE TREATMENT OF POLYCYCSTIC KIDNEY DISEASE AMERICAN CYANAMID COMPANY 2001-09-11 US disclosed