SCHEMBL7007537

SCHEMBL7007537

Brc1cc2c(cc1OCCC1CCCCN1)NCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
SSTR2 P30874 5/20 0.36
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
HRH3 Q9Y5N1 2/20 0.33
CHEK2 O96017 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
CHEK1 O14757 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HIF1A Q16665 1/20 0.32
PHLPP2 Q6ZVD8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7009169 0.74 CHEK2 (0.33) SSTR2PIM1PIM2CHEK2HSP90AA1
SCHEMBL7096511 0.74 HRH3 (0.54) HRH3SMN1; SMN2
SCHEMBL11449282 0.73 PIM1 (0.47) ALDH1A1PIM1PIM2CYP1A2CYP2D6
SCHEMBL8612335 0.72 HTR7 (0.44) ALDH1A1MAPTHRH3HTR2AHTR2C
SCHEMBL12491869 0.70 CHRNB4 (0.39) ALDH1A1MAPTCHEK1MKNK1
SCHEMBL11467927 0.69 CHRNB4 (0.50) ALDH1A1PIM1PIM2MKNK1SMN1; SMN2
SCHEMBL18152767 0.69 HTR2C (0.40) ALDH1A1MAPTPIM1PIM2HTR2A
SCHEMBL8615064 0.68 ALDH1A1 (0.37) ALDH1A1MAPTHRH3HTR2AHTR2C
SCHEMBL8617442 0.68 CHRNB4 (0.46)
SCHEMBL8613696 0.68 HRH3 (0.44) ALDH1A1MAPTHRH3HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309551-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002014273-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-21 WO disclosed