SCHEMBL7003896

SCHEMBL7003896

O=C(c1ccc(Cl)c(Cl)c1)C1CNCCC1(CCC(O)c1ccccc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 13/20 0.42
SLC6A2 P23975 12/20 0.39
SLC6A4 P31645 12/20 0.39
CYP2D6 P10635 1/20 0.39
KCNH2 Q12809 1/20 0.35
KMO O15229 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6995928 0.92 SLC6A3 (0.42) SLC6A3SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL7002582 0.81 SLC6A3 (0.48) SLC6A3SLC6A2SLC6A4CYP2D6
SCHEMBL7002761 0.76 LMNA (0.34)
SCHEMBL7002089 0.70 SLC6A2 (0.39) SLC6A3SLC6A2SLC6A4CYP2D6
SCHEMBL7003952 0.70 SLC6A4 (0.51) SLC6A3SLC6A2SLC6A4
SCHEMBL20399469 0.67 OPRM1 (0.47) SLC6A4
Hydrochloric Acid SCHEMBL20400820 0.67 OPRM1 (0.46) SLC6A4
SCHEMBL6995095 0.66 SLC6A3 (0.45) SLC6A3SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL7005083 0.66 SLC6A4 (0.41) SLC6A3SLC6A2SLC6A4
SCHEMBL6995034 0.66 SLC6A3 (0.38) SLC6A3SLC6A2SLC6A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed