SCHEMBL6995095

SCHEMBL6995095

O=C(c1ccc(Cl)c(Cl)c1)C1CNCCC1(O)CCc1ccc(Cl)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.45
SLC6A2 P23975 5/20 0.45
SLC6A4 P31645 5/20 0.45
CYP2D6 P10635 4/20 0.45
KCNH2 Q12809 3/20 0.39
KMO O15229 2/20 0.38
SIGMAR1 Q99720 1/20 0.37
UTS2R Q9UKP6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001083 0.83 ALDH1A1 (0.39) KCNH2
SCHEMBL7002582 0.73 SLC6A3 (0.48) SLC6A3SLC6A2SLC6A4CYP2D6
SCHEMBL5499282 0.72 SIGMAR1 (0.51) SLC6A2SLC6A4SIGMAR1
SCHEMBL6998084 0.70 HTR2A (0.38) SLC6A3SLC6A2SLC6A4
SCHEMBL13389380 0.69 SLC6A2 (0.44) SLC6A3SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL5499307 0.67 SIGMAR1 (0.49) SLC6A2SLC6A4KCNH2SIGMAR1
SCHEMBL6995928 0.67 SLC6A3 (0.42) SLC6A3SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL18519811 0.64 KMO (0.53) SLC6A3KMO
SCHEMBL21448810 0.64 KMO (0.53) SLC6A3KMO
SCHEMBL21448805 0.64 KMO (0.53) SLC6A3KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP disclosed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP disclosed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO disclosed