SCHEMBL7004059

SCHEMBL7004059

O=C(C1CNCCC1(CO)c1ccc(Cl)cc1Cl)C1CNCCC1(CO)c1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
UGCG Q16739 3/20 0.39
CYP3A4 P08684 4/20 0.38
KCNH2 Q12809 3/20 0.38
REN P00797 2/20 0.38
SLC6A4 P31645 13/20 0.37
SLC6A2 P23975 11/20 0.37
SLC6A3 Q01959 5/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005112 0.88 SLC6A3 (0.48) UGCGCYP3A4KCNH2RENSLC6A4
SCHEMBL7003952 0.79 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3
SCHEMBL7005083 0.72 SLC6A4 (0.41) RENSLC6A4SLC6A2SLC6A3
SCHEMBL7001284 0.71 LMNA (0.44) SLC6A3
SCHEMBL7002582 0.68 SLC6A3 (0.48) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL20978056 0.67 UGCG (0.45) UGCGCYP3A4SLC6A4SLC6A2SLC6A3
SCHEMBL1513518 0.67 DRD2 (0.58) UGCGSLC6A4SLC6A3
SCHEMBL21723004 0.66 SLC6A4 (0.57) SLC6A4SLC6A2SLC6A3
SCHEMBL7002089 0.65 SLC6A2 (0.39) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL7004831 0.64 REN (0.42) CYP3A4KCNH2RENSLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed