SCHEMBL7004077

SCHEMBL7004077

CCCCOc1c2cc(OC)c(OC)c(=O)c-2cn(CC(C)(C)C)c1C(=O)OCC

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 1/20 0.38
MAPT P10636 2/20 0.36
SIRT3 Q9NTG7 1/20 0.34
SIRT5 Q9NXA8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
TNF P01375 1/20 0.34
PDE4B Q07343 1/20 0.34
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003231 0.89 SLC6A5 (0.38) SLC6A5KDM4EALDH1A1
SCHEMBL7005350 0.86 SLC6A5 (0.38) SLC6A5MAPTSIRT3SIRT5KDM4E
SCHEMBL7564220 0.85 MAPT (0.38) MAPTSIRT3SIRT5KDM4EMEN1
SCHEMBL7006166 0.84 ESR1 (0.38) ALDH1A1
SCHEMBL7555960 0.82 TDP1 (0.38) MAPTKDM4EALDH1A1TNF
SCHEMBL7006171 0.77 ESR1 (0.34) SLC6A5MEN1ALDH1A1KMT2AGAA
SCHEMBL7001088 0.77 NPC1 (0.36) MAPTMEN1ALDH1A1KMT2A
SCHEMBL7007505 0.74 SLC6A5 (0.37) SLC6A5KDM4EALDH1A1KMT2AGAA
SCHEMBL7556201 0.74 MAPT (0.38) MAPTSIRT3SIRT5KDM4EMEN1
SCHEMBL5238999 0.72 TNF (0.40) SLC6A5MEN1ALDH1A1KMT2ATNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed