SCHEMBL7006166

SCHEMBL7006166

CCCCOc1c2cc(Cl)c(Cl)c(=O)c-2cn(CC(C)(C)C)c1C(=O)OCC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.38
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
ALDH1A1 P00352 1/20 0.33
POLB P06746 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
RAB9A P51151 1/20 0.31
ADRA1D P25100 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
NOTUM Q6P988 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
THRA P10827 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7555501 0.87 GPR35 (0.36) BAZ2BBAZ2AALDH1A1POLBADRA1D
SCHEMBL7006414 0.87 ESR1 (0.39) ESR1BAZ2BBAZ2AALDH1A1POLB
SCHEMBL7006924 0.84 CRHBP (0.44) ESR1ALDH1A1SMN1; SMN2CRHBPCRHR2
SCHEMBL7003687 0.84 ESR1 (0.37) ESR1BAZ2BBAZ2APOLBSMN1; SMN2
SCHEMBL7004077 0.84 SLC6A5 (0.38) ALDH1A1
SCHEMBL7000138 0.84 ESR1 (0.36) ESR1BAZ2BBAZ2AL3MBTL1
SCHEMBL7555960 0.83 TDP1 (0.38) ALDH1A1SMN1; SMN2NPC1CYP1A2CYP2C9
SCHEMBL7556806 0.83 BAZ2B (0.38) ESR1BAZ2BBAZ2AALDH1A1POLB
SCHEMBL7010259 0.82 ESR1 (0.39) ESR1BAZ2BBAZ2AALDH1A1SMN1; SMN2
SCHEMBL7003285 0.80 ESR1 (0.38) ESR1BAZ2BBAZ2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed