SCHEMBL7004172

SCHEMBL7004172

CC(=O)Nc1ccc(C2=C(c3ccc(S(N)(=O)=O)cc3)OC(C)(C)C2=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 11/20 0.58
CA2 P00918 11/20 0.58
CA12 O43570 8/20 0.58
CA9 Q16790 8/20 0.58
IDO1 P14902 1/20 0.49
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
PLK1 P53350 1/20 0.45
PTPN7 P35236 1/20 0.45
CA4 P22748 2/20 0.45
CA7 P43166 2/20 0.45
KMT2A Q03164 2/20 0.43
PKM P14618 1/20 0.43
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994970 0.84 CA2 (0.46) CA1CA2CA12CA9CA7
SCHEMBL7002958 0.83 CA2 (0.40) CA1CA2CA12CA9IDO1
SCHEMBL7003386 0.83 CA2 (0.49) CA1CA2CA12CA9CA7
SCHEMBL6999688 0.82 PTGS2 (0.60) CA1CA2CA12CA9PTPN7
SCHEMBL7002002 0.81 PTGS2 (0.56) CA1CA2CA12CA9CA4
SCHEMBL7000106 0.80 CA2 (0.53) CA1CA2CA12CA9CA4
SCHEMBL6998878 0.80 PTGS2 (0.57) CA1CA2CA12CA9CA4
SCHEMBL6992672 0.80 PTGS2 (0.51)
SCHEMBL6999710 0.79 CA2 (0.49) CA1CA2CA12CA9
SCHEMBL6994360 0.79 CHRNA7 (0.44) CA1CA2CA9ALDH1A1CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP claimed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US claimed
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP disclosed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US disclosed