SCHEMBL6994970

SCHEMBL6994970

CC(=O)c1ccc(C2=C(c3ccc(S(N)(=O)=O)cc3)OC(C)(C)C2=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.46
CA1 P00915 12/20 0.46
CA9 Q16790 12/20 0.46
CA12 O43570 11/20 0.46
PTGS2 P35354 5/20 0.44
CA14 Q9ULX7 10/20 0.42
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CYP2C19 P33261 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA5B Q9Y2D0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997640 0.89 PTGS2 (0.46) PTGS2
SCHEMBL7000178 0.87 CA2 (0.46) CA2CA1CA9CA12PTGS2
SCHEMBL6999843 0.86 CA1 (0.42) CA2CA1CA9CA12PTGS2
SCHEMBL7003386 0.86 CA2 (0.49) CA2CA1CA9CA12PTGS2
SCHEMBL6999688 0.85 PTGS2 (0.60) CA2CA1CA9CA12PTGS2
SCHEMBL6991749 0.85 PTGS2 (0.41) CA2CA1CA9CA12PTGS2
SCHEMBL6997787 0.85 PTGS2 (0.40) CA2CA1CA9CA12PTGS2
SCHEMBL7004172 0.84 CA1 (0.58) CA2CA1CA9CA12CA7
SCHEMBL7002002 0.84 PTGS2 (0.56) CA2CA1CA9CA12PTGS2
SCHEMBL6996692 0.84 RXRA (0.42) CA2CA1CA9CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP claimed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US claimed
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP claimed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO claimed
EP-1109799-B1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORP (KR) 2003-12-17 EP disclosed
US-6492416-B1 TREATING INFLAMMATION AND ASSOCIATED DISORDERS PACIFIC CORPORATION (KR) 2002-12-10 US disclosed
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP disclosed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO disclosed