SCHEMBL7004523

SCHEMBL7004523

O=c1[nH]ccn2c1cc1ccc(O)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
TYR P14679 1/20 0.38
CHEK1 O14757 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
GAA P10253 3/20 0.34
RAD51 Q06609 2/20 0.34
USP2 O75604 1/20 0.34
ALOX15 P16050 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PARP1 P09874 1/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 2/20 0.33
CA12 O43570 2/20 0.33
MCL1 Q07820 2/20 0.33
CA9 Q16790 2/20 0.33
CA1 P00915 1/20 0.33
GLA P06280 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001371 0.80 BRD4 (0.45) BRD4CHEK1CDK5CDK5R1PARP1
SCHEMBL7002739 0.80 GRIA1 (0.39) BRD4PARP1KDM4EDAOHTR2A
SCHEMBL7005550 0.80 CHEK1 (0.45) BRD4CHEK1KDM4EALDH1A1KMT2A
SCHEMBL7006748 0.80 BRD4 (0.45) BRD4CHEK1CDK5TYMSAURKA
SCHEMBL7005666 0.78 DAO (0.41) BRD4PARP1ALDH1A1DAOLMNA
SCHEMBL4751214 0.77 PARP1 (0.41) BRD4CHEK1GAAPARP1KDM4E
SCHEMBL7004919 0.76 MEN1 (0.42) BRD4NPSR1KDM4EMEN1ALDH1A1
SCHEMBL7006207 0.75 GRIA1 (0.41) ALOX15PARP1CA12CA9TDP1
SCHEMBL7007056 0.73 CES1 (0.38) KDM4EDAOL3MBTL1TDP2
SCHEMBL7003213 0.72 NSD2 (0.50) CHEK1MEN1KMT2ACA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1200439-B1 1,2-DIHYDRO-1-OXO-PARAZINO(1,2-A) INDOLE DERIVATIVES NOVUSPHARMA SPA (IT) 2003-06-25 EP disclosed