SCHEMBL7005550

SCHEMBL7005550

O=c1[nH]ccn2c1cc1ccc(Cl)cc12

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.45
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
HPGD P15428 1/20 0.39
BRD4 O60885 1/20 0.38
CMA1 P23946 1/20 0.38
AHR P35869 1/20 0.38
TDP2 O95551 3/20 0.37
DAO P14920 2/20 0.36
PTPN1 P18031 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
EGFR P00533 1/20 0.35
KMT2A Q03164 1/20 0.35
F11 P03951 1/20 0.35
KMO O15229 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001371 0.80 BRD4 (0.45) CHEK1ALDH1A1KDM4ECYP1A2BRD4
SCHEMBL7006748 0.80 BRD4 (0.45) CHEK1BRD4AHR
SCHEMBL7002739 0.80 GRIA1 (0.39) KDM4EBRD4AHRDAOHTR2A
SCHEMBL7005666 0.78 DAO (0.41) ALDH1A1CYP1A2BRD4DAO
SCHEMBL4751214 0.77 PARP1 (0.41) CHEK1ALDH1A1KDM4EHPGDBRD4
SCHEMBL7004919 0.76 MEN1 (0.42) ALDH1A1KDM4ECYP1A2HPGDBRD4
SCHEMBL7006207 0.75 GRIA1 (0.41) CYP1A2DAO
SCHEMBL7007056 0.73 CES1 (0.38) KDM4ETDP2DAO
SCHEMBL7003383 0.72 TDP2 (0.39) BRD4TDP2DAOPTPN1HTR2A
SCHEMBL7003213 0.69 NSD2 (0.50) CHEK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1200439-B1 1,2-DIHYDRO-1-OXO-PARAZINO(1,2-A) INDOLE DERIVATIVES NOVUSPHARMA SPA (IT) 2003-06-25 EP disclosed