SCHEMBL7004530

SCHEMBL7004530

CC(=O)Oc1c2ccsc2cc2sccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GAA P10253 2/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
ABCB11 O95342 1/20 0.39
BACE1 P56817 1/20 0.38
PREP P48147 3/20 0.36
CELA1 Q9UNI1 2/20 0.36
TOP1 P11387 1/20 0.36
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003660 0.86 TUBB4A (0.52) HTTKDM4EHSD17B10GAATP53
SCHEMBL6993194 0.85 TUBB4A (0.37) HTTKDM4EHSD17B10GAATP53
SCHEMBL6001768 0.78 ALDH1A1 (0.51) HTTKDM4EGAAMAPTTUBB4A
SCHEMBL7519724 0.77 HDAC3 (0.38) HTTKDM4EHSD17B10GAATP53
SCHEMBL10682692 0.74 CSNK2A2 (0.37) KDM4EHSD17B10GAAMAPTCSNK2A2
SCHEMBL644865 0.74 KDM4E (0.53) HTTKDM4EHSD17B10GAATP53
SCHEMBL11053213 0.73 KDM4E (0.44) HTTKDM4EHSD17B10GAAMAPT
SCHEMBL5742360 0.71 MAPK1 (0.44) HTTKDM4EHSD17B10GAAMAPT
SCHEMBL8148551 0.69 KDM4E (0.34) HTTKDM4EHSD17B10GAAMAPT
SCHEMBL10903229 0.69 GPR35 (0.49) KDM4EHSD17B10GAATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093456-B1 NAPHTHO- AND DIHYDROBENZO-THIOPHENE DERIVATIVES AS CYTOTOXIC ANTITUMOR AGENTS UNIV NORTH CAROLINA (US) 2003-12-17 EP disclosed
US-6337346-B1 BENZODITHIOPHENE DERIVATIVES UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2002-01-08 US disclosed
EP-1093456-A2 NAPHTHO- AND DIHYDROBENZO-THIOPHENE DERIVATIVES AS CYTOTOXIC ANTITUMOR AGENTS UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2001-04-25 EP disclosed
US-6174913-B1 TREATING TUMOR BY ADMINISTERING COMPOUNDS E.G.:2-ACETYL-NAPHTHO(2,3-B)THIOPHENE-4,9-DIONE; 2,7-DIACETYL-NAPHTHO(2,3-B)THIOPHENE-4,9-DIONE THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2001-01-16 US disclosed
WO-1999062909-A9 NAPHTHO- AND DIHYDROBENZO-THIOPHENE DERIVATIVES AS CYTOTOXIC ANTITUMOR AGENTS UNIV NORTH CAROLINA (US) 2000-04-27 WO disclosed
WO-1999062909-A2 NAPHTHO- AND DIHYDROBENZO-THIOPHENE DERIVATIVES AS CYTOTOXIC ANTITUMOR AGENTS UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-12-09 WO disclosed