SCHEMBL7004599

SCHEMBL7004599

CCc1cccc2c(C(=O)OC(C)(C)C)c[nH]c12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.62
LMNA P02545 3/20 0.62
HTT P42858 1/20 0.62
MEN1 O00255 5/20 0.57
KMT2A Q03164 5/20 0.57
MAPT P10636 5/20 0.57
RAB9A P51151 2/20 0.57
MAPK1 P28482 2/20 0.57
NPC1 O15118 1/20 0.57
CASP3 P42574 1/20 0.57
SENP7 Q9BQF6 1/20 0.57
NPSR1 Q6W5P4 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NR4A2 P43354 2/20 0.49
TSHR P16473 1/20 0.48
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
UBE2N P61088 1/20 0.47
USP2 O75604 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1037516 0.82 NR4A2 (0.50) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL1466935 0.81 ALDH1A1 (0.74) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL16453789 0.78 ALDH1A1 (0.80) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL5943223 0.77 ALDH1A1 (0.68) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL16453792 0.77 ALDH1A1 (0.68) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL6196294 0.75 NR4A2 (0.39) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL10675123 0.75 ALDH1A1 (0.62) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL6684094 0.75 NR4A2 (0.69) ALDH1A1LMNAHTTMEN1KMT2A
SCHEMBL1759590 0.74 NR4A2 (0.47) MEN1KMT2AMAPTNR4A2
SCHEMBL22492440 0.74 CLEC4M (0.80) ALDH1A1LMNAHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1245405-C Piperazine derivatives HOFFMANN LA ROCHE (CH) 2006-03-15 CN disclosed
CN-1529706-A Piperazine derivatives - 2004-09-15 CN disclosed
EP-1370561-A2 TETRAHYDRO-PYRAZINO[1,2-A]INDOLES FOR THE TREATMENT OF CENTRAL NERVOUS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2003-12-17 EP disclosed
EP-1325008-A1 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-07-09 EP disclosed
WO-2002072584-A2 TETRAHYDRO-PYRAZINO (1,2-A) INDOLES FOR THE TREATMENT OF CENTRAL NERVOUS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2002-09-19 WO disclosed
WO-2002010169-A1 PIPERAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-02-07 WO disclosed