SCHEMBL7005299

SCHEMBL7005299

O=C(NCC(=O)c1cn(CCCN2C(=O)c3ccccc3C2=O)c2ccccc12)Nc1cccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.54
CNR1 P21554 3/20 0.54
KDM4E B2RXH2 3/20 0.43
HSD17B10 Q99714 2/20 0.43
GSK3B P49841 1/20 0.42
EPHX1 P07099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7009092 0.84 MAPT (0.43) CNR2CNR1
SCHEMBL7010065 0.82 CNR2 (0.42) CNR2CNR1KDM4E
SCHEMBL7007071 0.78 CAMK2D (0.47) CNR2CNR1
SCHEMBL7250031 0.75 MAPT (0.55) KDM4EHSD17B10
SCHEMBL8837853 0.75 SMN1; SMN2 (0.60) CNR2CNR1
SCHEMBL29362081 0.70 CNR2 (1.00) CNR2CNR1
SCHEMBL9238742 0.70 SMN1; SMN2 (0.55) CNR2CNR1
SCHEMBL29019173 0.70 CNR2 (0.78) CNR2CNR1
SCHEMBL8837847 0.68 CNR2 (0.43) CNR2CNR1
SCHEMBL17943658 0.68 CNR2 (0.41) CNR2CNR1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030134886-A1 Pharmaceutically active compounds ASTRAZENECA AB, A SWEDISH CORPORATION 2003-07-17 US disclosed
EP-1042317-B1 Indole derivatives as PKC-inhiboitors ASTRAZENECA AB (SE) 2003-05-14 EP disclosed
US-6492409-B1 SUCH AS 5-(1-(3-AMINOPROPYL)-3-INDOLYL)-1-(3-INDOLYL)-1,3-DIHYDROIMIDAZOL-2-ONE; PROTEIN KINASE C INHIBITORS; HIGH SOLUBILITY; REDUCED COLOR; TREATING INFLAMMATORY AND/OR IMMUNOLOGICAL DISORDERS ASTRAZENECA AB (SE) 2002-12-10 US disclosed
US-6337342-B1 ARYLIMIDAZOLONE DERIVATIVES ASTRAZENECA AB (SE) 2002-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030134886-A1 Pharmaceutically active compounds HTR3C, HTR6, CNR1 CNR2 30/4885CNR1 3/4885KDM4E 1063/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.