SCHEMBL7005305

SCHEMBL7005305

CC(C)(C)n1cc(-c2ccc(-c3ccccc3)cc2)c(C#N)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
LMNA P02545 2/20 0.44
ADORA1 P30542 8/20 0.42
KDM4E B2RXH2 5/20 0.41
HPGD P15428 3/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPK1 P28482 2/20 0.41
GAA P10253 1/20 0.41
ADORA2A P29274 6/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
LCK P06239 1/20 0.38
SRC P12931 1/20 0.38
KDR P35968 1/20 0.38
TEK Q02763 1/20 0.38
MEN1 O00255 1/20 0.38
PIM1 P11309 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GRM6 O15303 1/20 0.37
CA12 O43570 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6862112 0.88 LCK (0.53) ALDH1A1LMNAADORA1KDM4EADORA2A
SCHEMBL7008781 0.88 PLA2G1B (0.40) ALDH1A1LMNAADORA1KDM4EHPGD
SCHEMBL6250271 0.87 SRC (0.47) ALDH1A1LMNAADORA1KDM4EHPGD
SCHEMBL7009014 0.85 CA12 (0.36) ALDH1A1LMNAADORA1KDM4EHPGD
SCHEMBL3715556 0.85 CA12 (0.50) ALDH1A1LMNAADORA1KDM4EHPGD
SCHEMBL7008786 0.82 ALDH1A1 (0.37) ALDH1A1LMNAADORA1KDM4EHPGD
SCHEMBL8508548 0.80 LCK (0.53) ALDH1A1ADORA1KDM4EHPGDADORA2A
SCHEMBL20162762 0.72 CA12 (0.46) ALDH1A1LMNAADORA1KDM4EHPGD
SCHEMBL7835925 0.72 CA12 (0.54) ALDH1A1LMNAADORA1KDM4EHPGD
SCHEMBL7008096 0.71 POLB (0.46) ALDH1A1LMNAADORA1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970084-B1 PYRROLO 2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AG (DE) 2003-06-04 EP disclosed
EP-0970084-A1 PYRROLO 2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-01-12 EP disclosed
US-6001839-A Substituted 4-amino-7H-pyrrolo [2,3,-d]-pyrimidines as PTK inhibitors BASF AKTIENGESELLSCHAFT (DE) 1999-12-14 US disclosed
WO-1998041525-A1 PYRROLO[2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-09-24 WO disclosed