SCHEMBL7008781

SCHEMBL7008781

CC(C)(C)n1cc(-c2ccc(Sc3ccccc3)cc2)c(C#N)c1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G1B P04054 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
ALDH1A1 P00352 8/20 0.37
LMNA P02545 3/20 0.37
L3MBTL1 Q9Y468 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
KDM4E B2RXH2 6/20 0.35
HPGD P15428 5/20 0.35
GAA P10253 1/20 0.35
MAPK1 P28482 1/20 0.35
LCK P06239 1/20 0.35
SRC P12931 1/20 0.35
KDR P35968 1/20 0.35
TEK Q02763 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
CYP1A2 P05177 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005305 0.88 ALDH1A1 (0.44) ALDH1A1LMNAL3MBTL1KDM4EHPGD
SCHEMBL6862112 0.82 LCK (0.53) MAOAALDH1A1LMNAL3MBTL1KDM4E
SCHEMBL6250271 0.81 SRC (0.47) ALDH1A1LMNATDP1KDM4EHPGD
SCHEMBL3715556 0.80 CA12 (0.50) ALDH1A1LMNAL3MBTL1TDP1KDM4E
SCHEMBL7009014 0.80 CA12 (0.36) ALDH1A1LMNAKDM4EHPGDGAA
SCHEMBL8508548 0.74 LCK (0.53) ALDH1A1KDM4EHPGDLCKSRC
SCHEMBL7008786 0.74 ALDH1A1 (0.37) ALDH1A1LMNAKDM4EHPGDGAA
SCHEMBL7004986 0.69 SRC (0.71) LCKSRCKDRTEK
SCHEMBL20162762 0.68 CA12 (0.46) ALDH1A1LMNAL3MBTL1TDP1KDM4E
SCHEMBL7008096 0.66 POLB (0.46) ALDH1A1LMNAL3MBTL1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970084-B1 PYRROLO 2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AG (DE) 2003-06-04 EP disclosed
EP-0970084-A1 PYRROLO 2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-01-12 EP disclosed
US-6001839-A Substituted 4-amino-7H-pyrrolo [2,3,-d]-pyrimidines as PTK inhibitors BASF AKTIENGESELLSCHAFT (DE) 1999-12-14 US disclosed
WO-1998041525-A1 PYRROLO[2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-09-24 WO disclosed