SCHEMBL7005680

SCHEMBL7005680

COc1c(-c2ccncc2)c(-c2ncnn2C)nn2c(-c3ccon3)nnc12

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.34
HSD17B10 Q99714 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA3 P34903 1/20 0.31
APAF1 O14727 1/20 0.30
HPGD P15428 1/20 0.30
RECQL P46063 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001199 0.87 HPGD (0.36) LRRK2HSD17B10NPC1GABRG2GABRB3
SCHEMBL7003645 0.85 LRRK2 (0.32) LRRK2GABRG2GABRB3
SCHEMBL7002972 0.70 HPGD (0.36) LRRK2HSD17B10NPC1RAB9AGABRG2
SCHEMBL7001541 0.69 LRRK2 (0.32) LRRK2GABRG2GABRB3
SCHEMBL7002883 0.68 GABRA1 (0.32) LRRK2GABRG2GABRB3GABRA3
SCHEMBL7002461 0.67 GABRA1 (0.33) LRRK2GABRG2GABRB3GABRA3
SCHEMBL2656994 0.66 GABRG2 (0.65) GABRG2GABRB3GABRA3
SCHEMBL7002447 0.64 GABRA1 (0.35) LRRK2NPC1RAB9AGABRG2GABRB3
SCHEMBL7482590 0.63 GABRA1 (0.52) GABRG2GABRB3GABRA3
SCHEMBL7208541 0.62 GABRG2 (0.46) GABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107967-B1 TRIAZOLOPYRIDAZINE DERIVATIVES FOR ENHANCING COGNITION MERCK SHARP & DOHME (GB) 2003-05-14 EP claimed