SCHEMBL7006291

SCHEMBL7006291

CCOC(=O)c1[nH]c2cc(O)cc(Cc3ccc(OC)cc3)c2c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.47
ALDH1A1 P00352 8/20 0.47
HPGD P15428 7/20 0.47
MAPT P10636 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
LMNA P02545 5/20 0.45
HSD17B10 Q99714 4/20 0.45
HTT P42858 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
ALOX5 P09917 1/20 0.43
ALOX15 P16050 2/20 0.42
KMT2A Q03164 5/20 0.42
NQO2 P16083 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9023820 0.85 MAPT (0.46) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL7004585 0.73 MAPT (0.41) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL7006235 0.69 ALDH1A1 (0.43) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL6859385 0.69 HTR6 (0.61) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL8902071 0.69 KDM4E (0.42) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL18796724 0.68 PDE3B (0.76) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL18531909 0.67 GAA (0.63) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL3954170 0.67 ALDH1A1 (0.47) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL38665015 0.66 ALDH1A1 (0.78) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL6598094 0.66 ALDH1A1 (0.58) KDM4EALDH1A1HPGDMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1341761-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2003-09-10 EP disclosed
WO-2002030895-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-η BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-18 WO disclosed