SCHEMBL7006366

SCHEMBL7006366

CCOC(=O)Oc1c(-c2ccncc2)c(-c2cccs2)n2c1CCC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
KCNK3 O14649 1/20 0.37
ALDH1A1 P00352 8/20 0.37
HPGD P15428 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HIF1A Q16665 1/20 0.37
MAPT P10636 2/20 0.36
GAA P10253 1/20 0.36
KEAP1 Q14145 1/20 0.36
KDM4E B2RXH2 3/20 0.35
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
ALOX5 P09917 1/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 3/20 0.35
PKM P14618 1/20 0.35
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
CA1 P00915 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013150 0.93 KMT2A (0.40) KMT2AMEN1KCNK3ALDH1A1HPGD
SCHEMBL7006701 0.86 ALOX5 (0.41) KMT2AMEN1ALDH1A1NPSR1KDM4E
SCHEMBL7009127 0.85 SMN1; SMN2 (0.38) ALDH1A1HPGDNPSR1MAPTGAA
SCHEMBL6294039 0.85 ALDH1A1 (0.47) KMT2AMEN1KCNK3ALDH1A1HPGD
SCHEMBL6294501 0.83 KCNK3 (0.48) KMT2AMEN1KCNK3ALDH1A1HPGD
SCHEMBL7012237 0.83 RIPK3 (0.45) KMT2A
SCHEMBL7008536 0.83 RIPK3 (0.45) KMT2A
SCHEMBL7006189 0.80 RIPK3 (0.44) KMT2A
SCHEMBL7011496 0.78 NPSR1 (0.38) ALDH1A1HPGDNPSR1MAPTGAA
SCHEMBL7010615 0.77 MAPK14 (0.44) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252163-B1 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2003-09-24 EP disclosed